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2022
 G. Loren, I. Espuny, A. Llorente, C. Donoghue, X. Verdaguer, R. Gomis, A. Riera Design and optimization of oestrogen receptor PROTACs based on 4-hydroxytamoxifen.
Eur. J. Med. Chem.,
243, 114770 (2022).

 P. Rojo, M. Molinari, A. Cabré, C. García-Mateos, A. Riera, X. Verdaguer Iridium-Catalyzed Asymmetric Hydrogenation of 2,3-Diarylallyl Amines with a Threonine-Derived P-Stereogenic Ligand for the Synthesis of Tetrahydroquinolines and Tetrahydroisoquinolines.
Angew. Chem. Int. Ed.,
0, e202204300 (2022).

 Enric Ros, M. Bellido, J.A. Matarin, A. Gallen, M. Mart´ınez, L. Rodrıguez, X. Verdaguer, L. Ribas de Pouplana, A. Riera Amino acids with fluorescent tetrazine ethers as bioorthogonal handles for peptide modification.
RSC Advances,
12, 14321 (2022).

 A. Cabré, X. Verdaguer, A. Riera Recent Advances in the Enantioselective Synthesis of Chiral Amines via Transition Metal-Catalyzed Asymmetric Hydrogenation.
Chem. Rev. ,
122, 269−339 (2022).


2021
 P. Rojo, A. Riera, X. Verdaguer BOM-Phosphinite as an Electrophilic P‑Stereogenic Transfer Reagent for the Synthesis of Bulky Phosphines: Synthesis of tert-Butyl(3,5-di-tert-butylphenyl)BisP*.
Org. Lett.,
23, 4802-4806 (2021).

 A. Rol et.al Structure-based design of a Cortistatin analogue with immunomodulatory activity in models of inflammatory bowel disease.
Nature. Commun. ,
12, 1869 (2021).


2020
 E. Ros, A. Prades, D. Forson,J. Smyth, X. Verdaguer, L. Ribas de Pouplana, A. Riera Synthesis of 3-alkyl-6-methyl-1,2,4,5-tetrazines via a Sonogashira-type cross-coupling reaction.
Chem. Commun. ,
56, 11086-11089 (2020).
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 A. Cabré, M. Garçon, A. Gallén, L. Grisoni, A. Grabulosa, X. Verdaguer, A. Riera Iridium-Catalyzed Asymmetric Isomerization of Primary Allylic Alcohols Using MaxPHOX Ligands: Experimental and Theoretical Study.
Chem. Cat. Chem. ,
12, 4112-4120 (2020).
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 A. Cabré, S. Rafael, G. Sciortino, G. Ujaque, X. Verdaguer, A. Lledós, A. Riera Catalytic Regioselective Isomerization of 2,2-Disubstituted Oxetanes to Homoallylic Alcohols.
Angew. Chem Int. Ed.,
59, 7521-7527 (2020).
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 E. Ros, M. Bellido, X. Verdaguer, L. Ribas de Pouplana, A. Riera Synthesis and Application of 3‑Bromo-1,2,4,5-Tetrazine for Protein Labeling to Trigger Click-to-Release Biorthogonal Reactions.
Bioconjugate Chem. ,
31, 933-938 (2020).
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